平安! 发表于 2011-11-9 19:57
/ n7 J ^1 C7 a$ ~9 ^Pazopanib (100 mg/kg/day free base equivalent)
% S0 t4 ^, E* | 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
7 t$ R. R# [. p4 N7 h搜索了一下,原料一大堆。
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0 a- A$ }: a& o对不起!100mg/kg是用于移植瘤的,我弄错了。6 ?/ j c7 i+ h6 G5 \) b
2 t5 ]$ B) J9 }! C' ]以下是正版说明书的推荐用量。
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--------------------- DOSAGE AND ADMINISTRATION ---------------- h1 q! l, a8 n+ x. @* ~
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) ) @# j4 W+ U @' @3 R9 l. L- L
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
3 j! H2 Y1 q: U" j: x+ V---------------------DOSAGE FORMS AND STRENGTHS --------------
5 S* @' ?) _( f2 ^200 mg tablets. (3)
& Q$ ]+ W* D' E3 D7 [# [, f-------------------------------CONTRAINDICATIONS------------------------ |